Screening of a Custom-Designed Acid Fragment Library Identifies 1-Phenylpyrroles and 1-Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity
Mahy W., Patel M., Steadman D., Woodward HL., Atkinson BN., Svensson F., Willis NJ., Flint A., Papatheodorou D., Zhao Y., Vecchia L., Ruza RR., Hillier J., Frew S., Monaghan A., Costa A., Bictash M., Walter MW., Jones EY., Fish PV.