Screening of a Custom-Designed Acid Fragment Library Identifies 1-Phenylpyrroles and 1-Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity

Mahy W., Patel M., Steadman D., Woodward HL., Atkinson BN., Svensson F., Willis NJ., Flint A., Papatheodorou D., Zhao Y., Vecchia L., Ruza RR., Hillier J., Frew S., Monaghan A., Costa A., Bictash M., Walter MW., Jones EY., Fish PV.

DOI

10.1021/acs.jmedchem.0c00660

Type

Journal article

Journal

Journal of Medicinal Chemistry

Publisher

American Chemical Society (ACS)

Publication Date

18/08/2020

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